Papers 2003

2,4-Diaminopyrimidines as Inhibitors of Leishmanial and Trypanosomal Dihydrofolate Reductase. Pez, D.; Leal, I.; Zuccotto, F.; Boussard, C.; Brun, R.; Croft, S. L.; Yardley, V.; Ruiz Perez, L. M.; Gonzalez Pacanowska, D.; Gilbert, I. H. Bioorg. Med. Chem., 2003, 11, 4693-4711.  link to journal abstract in pubmed  link to the journal where paper was published

Azasterols as Inhibitors of Sterol 24-Methyltransferase in Leishmania and Trypanosoma cruzi. Magaraci, F.; Jimenez Jimenez, C.; Rodrigues, C.; Rodrigues, J. C. F.; Vianna Braga, M.; Yardley, V.; de Luca-Fradley, K.; Croft, S. L.; de Souza, W.; Ruiz-Perez, L. M.; Urbina, J.; Gonzalez Pacanowska,  D.; Gilbert, I. H. J. Med. Chem., 2003, 46, 4714-4727.  link to journal abstract in pubmed  link to the journal where paper was published

Anti-Plasmodial activity of a series of 1,3,5 triazine substituted polyamines. Klenke, B.; Barrett,  M. P.; Brun, R.; Gilbert, I. H. J. Antimicrob. Chemoth., 2003, 52 , 290-293.  link to journal abstract in pubmed  link to the journal where paper was published

Synthesis and biological evaluation of substrate-based inhibitors of 6-phosphogluconate dehydrogenase as potential drugs against African Trypanosomiasis. Dardonville, C.; Rinaldi, E.; Hanau, S.; Barrett, M. P.; Brun, R.; Gilbert, I. H. Bioorg. Med. Chem., 2003, 11, 3205-3214.  link to journal abstract in pubmed  link to the journal where paper was published

Synthesis and Evaluation of Analogues of Congo Red as Potential Compounds against Transmissible Spongiform Encephalopathies. Rudyk, H.; Knaggs, M. H.; Vasiljevic, S.; Hope, J.; Birkett, C.; Gilbert, I. H. Eur. J. Med. Chem., 2003, 38, 567-579.  link to journal abstract in pubmed  link to the journal where paper was published

Synthesis of (R)-2-methyl-4-deoxy and (R)-2-methyl-4, 5-dideoxy analogues of 6-phosphogluconate as potential inhibitors of 6-phosphogluconate dehydrogenase. Dardonville, C.; Gilbert, I. H. Org. Biomol. Chem., 2003, 1, 552-559.  link to journal abstract in pubmed  link to the journal where paper was published

In vitro cell-free conversion of bacterial recombinant PrP to PrPres as a model for conversion. Kirby, L.; Birkett, C. R.; Rudyk, H.; Gilbert, I. H.; Hope, J. J. Gen. Virol., 2003, 84 , 1013-1020 .  link to journal abstract in pubmed  link to the journal where paper was published

Solid-Phase Synthesis of Diamine and Polyamine Amino Acid Derivatives as HIV-1 Tat-TAR Binding Inhibitors. Jimenez Bueno, G.; Klimkait, T.; Gilbert, I. H.; Simons, C. Bioorg. Med. Chem., 2003, 11, 87-94.  link to journal abstract in pubmed  link to the journal where paper was published

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