Design, Synthesis and Evaluation of Inhibitors of Trypanosomal and Leishmanial Dihydrofolate Reductase. Chowdhury, S. F.; Bernier Villamor, V.; Hurtado Guerrero, R.; Leal, I.; Brun, R.; Croft, S. L.; Goodman, J. M.; Maes, L.; Ruiz-Perez, L. M.; Gonzalez Pacanowska, D.; Gilbert, I. H. J. Med. Chem., 1999, 42 , 4300-4312.
The Design and Synthesis of Lipophilic, Phosphoramidate d4T-MP Prodrugs Expressing High Potency Against HIV in Cell Culture: Structural Determinants for in vitro Activity and QSAR. Siddiqui, A.; McGuigan, C.; Gilbert, I.H.; Ballatore, C.; Zuccotto, F.; De Clercq, E.; Balzarini, J. J. Med. Chem., 1999,42, 4122-4128.
Inhibitors of Protease-Resistant Prion Formation. Gilbert I. H.; Rudyk, H.; International Antiviral News, 1999, 7, 78-82.
The Structure-Based Design And Synthesis Of Selective Inhibitors of Trypanosoma cruzi Dihydrofolate Reductase. Zuccotto, F.; Brun, R.; Gonzalez Pacanowska, D.; Ruiz Perez, L. M.; Gilbert, I. H. Bioorg. Med. Chem. Lett., 1999, 9, 1463-1468.
General Synthesis of 3-Phosphorylated myo-Inositol Phospholipids and their Derivatives. Painter, G. F.; Grove, S. J. A.; Gilbert, I. H.; Holmes, A. B.; Raithby, P. R.; Hill, M. L.; Hawkins, P. T.; Stephens, L. R. J. Chem. Soc., Perk. T 1, 1999, 923-936.
Design And Synthesis Of Bio-Isosteres Of Thymidine Triphosphate. Goldring, A. O.; Balzarini, J.; Gilbert, I. H. Bioorg. Med. Chem. Lett., 1998, 8, 1211-1215.
An Approach To Use An Unusual Adenosine Transporter To Selectively Deliver Polyamine Analogues To Trypanosomes. Tye, C.-K.; Kasinathan, G.; Barrett, M. P.; Brun, R.; Doyle, V. E.; Fairlamb, A. H.; Weaver R.; Gilbert, I. H. Bioorg. Med. Chem. Lett., 1998, 8, 811-816.
Electrospray Mass Spectrometry For Assay of Erythromycin A Extracted From Fermentation Liquor. Morgan, J.; Rowlands, R. T.; Joyce-Menekse, M. E.; Gilbert, I. H.; Lloyd, D. Biotechnol. Tech., 1998, 12, 435-438.
Dihydrofolate Reductase: a Potential Drug Target in Trypanosomes and Leishmania. Zuccotto, F.; Martin, A. C. R.; Laskowski, R. A.; Thornton, J. M.; Gilbert, I. H. J. Comput. Aid. Mol. Des., 1998, 12, 241-257.
Versatile Synthesis of myo-Inositol Phospholipid Precursors. Grove, S. J. A.; Gilbert, I. H.; Holmes, A. B.; Painter, G. F.; Hill, M. L. Chem. Commun., 1997, 1633-1634.
The Design and Synthesis of Nucleoside Triphosphate Isosteres as Potential Inhibitors of HIV Reverse Transcriptase. R. Weaver, I. H. Gilbert, Tetrahedron, 1997, 53, 5537-5562.
Lipophilic Bioisosteres of Nucleoside Triphosphates. Goldring, A. O.; Gilbert, I. H.; Mahmood, N.; Balzarini, J. Bioorg. Med. Chem. Lett., 1996, 6, 2411-2416.
Isosteres of Nucleoside Triphosphates. Weaver, R.; Gilbert, I. H.; Mahmood, N.; Balzarini, J. Bioorg. Med. Chem. Lett., 1996, 6, 2405-2410.
Synthesis of β -Keto and αβ -Unsaturated N-Acetylcysteamine Thioesters. Gilbert, I. H.; Ginty, M.; O’Neill, J. A.; Simpson, T. J.; Staunton J.; Willis C. L. Bioorg. Med. Chem. Lett, 1995, 5, 1587-1590.
Imidazolines as Amide Bond Replacements. Gilbert, I. H.; Rees, D. C.; Crockett, A. K.; Jones, R. C. F. Tetrahedron, 1995, 51, 6315-6335.
Synthesis of a Homochiral Alpha, Alpha-Disubstituted Alpha, Beta-Diamino-Acid. Jones, R. C. F.; Crockett, A. K.; Rees D. C.; Gilbert, I. H. Tetrahedron-Asymmetr., 1994, 5, 1661-1664.
Lewis Acid Catalysed rearrangements of myo-inositol orthoformate derivatives. Gilbert, I. H. Holmes, A. B.; Pestchanker, M. J.; Young, R. C. Carbohyd. Res., 1992, 234, 117-130.
Amide bond replacements: incorporation of a 2,5,5-trisubstituted imidazoline into dipeptides and into a CCK-4 derivative. Gilbert, I. H.; Rees, D. C.; Richardson, R. S. Tetrahedron Lett., 1991, 32, 2277-2280.
Synthesis of Protected myo-Inositols. Gilbert, I. H.; Holmes, A. B.; Young, R. C. Tetrahedron Lett., 1990, 31, 2633-2634.