Prioritization of Molecular Targets for Antimalarial Drug Discovery
Barbara Forte, Sabine Ottilie, Andrew Plater, Brice Campo, Koen J. Dechering, Francisco Javier Gamo, Daniel E. Goldberg, Eva S. Istvan, Marcus Lee, Amanda K. Lukens, Case W. McNamara, Jacquin C. Niles, John Okombo, Charisse Flerida A. Pasaje, Miles G. Siegel, Dyann Wirth, Susan Wyllie, David A. Fidock, Beatriz Baragaña, Elizabeth A. Winzeler, and Ian H. Gilbert ACS Infectious Diseases 2021 7 (10), 2764-2776
DOI: 10.1021/acsinfecdis.1c00322
Mycobacterium tuberculosis Phe-tRNA synthetase: structural insights into tRNA recognition and aminoacylation
Karolina Michalska, Robert Jedrzejczak, Jacek Wower, Changsoo Chang, Beatriz Baragaña, Ian H Gilbert, Barbara Forte, Andrzej Joachimiak
Nucleic Acids Research, Volume 49, Issue 9, 21 May 2021, 5351–5368 https://doi.org/10.1093/nar/gkab272
MalDA, Accelerating Malaria Drug Discovery
Tuo Yang, Sabine Ottilie, Eva S Istvan, Karla P Godinez-Macias, Amanda K Lukens, Beatriz Baragaña, Brice Campo, Chris Walpole, Jacquin C Niles, Kelly Chibale, Koen J Dechering , Manuel Llinás , Marcus C S Lee, Nobutaka Kato, Susan Wyllie, Case W McNamara, Francisco Javier Gamo, Jeremy Burrows, David A Fidock, Daniel E Goldberg, Ian H Gilbert, Dyann F Wirth, Elizabeth A Winzeler, Malaria Drug Accelerator Consortium.
Trends Parasitol. 2021 , Volume 37, Issue 6, 493-507, June 01, 2021 DOI: 10.1016/j.pt.2021.01.009
Chemogenomics identifies acetyl-coenzyme A synthetase as a target for malaria treatment and prevention
Robert L Summers RL, Charisse Flerida A Pasaje CFA, Joao P Pisco JP, Josefine Striepen J, Madeline R Luth MR, Krittikorn Kumpornsin K, Emma F Carpenter EF, Justin T Munro JT, De Lin , Andrew Plater A, Avinash S Punekar AS, Andrew M Shepherd AM, Sharon M Shepherd SM, Manu Vanaerschot M, James M Murithi JM, Kelly Rubiano K, Aslı Akidil A, Sabine Ottilie S, Nimisha Mittal N, A Hazel Dilmore AH, Madalyn Won M, Rebecca E K Mandt REK, Kerry McGowen K, Edward Owen E, Chris Walpole C, Manuel Llinás M, Marcus C S Lee MCS, Elizabeth A Winzeler EA, David A Fidock DA, Ian H Gilbert IH, Dyann F Wirth DF, Jacquin C Niles JC, Beatriz Baragaña B, Amanda K Lukens AK
Cell chemical biology (2021), https://doi.org/10.1016/j.chembiol.2021.07.010
Lysyl-tRNA synthetase as a drug target in malaria and cryptosporidiosis
Beatriz Baragaña, Barbara Forte, Ryan Choi, Stephen Nakazawa Hewitt et al.
PNAS April 2, 2019 116 (14) 7015-7020; first published March 20, 2019; https://doi.org/10.1073/pnas.1814685116