{"id":704,"date":"2013-09-17T21:14:53","date_gmt":"2013-09-17T21:14:53","guid":{"rendered":"http:\/\/blog.dundee.ac.uk\/ian-gilbert\/?page_id=704"},"modified":"2013-12-20T13:15:31","modified_gmt":"2013-12-20T13:15:31","slug":"papers-pre-2000","status":"publish","type":"page","link":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/papers-pre-2000\/","title":{"rendered":"Papers pre-2000"},"content":{"rendered":"

Design, Synthesis and Evaluation of Inhibitors of Trypanosomal and Leishmanial Dihydrofolate Reductase. Chowdhury, S. F.; Bernier Villamor, V.; Hurtado Guerrero, R.; Leal, I.; Brun, R.; Croft, S. L.; Goodman, J. M.; Maes, L.; Ruiz-Perez, L. M.; Gonzalez Pacanowska, D.; Gilbert, I. H. J. Med. Chem., 1999, 42 , 4300-4312.\u00a0 \"link<\/a>\u00a0 \"link<\/a><\/p>\n

The Design and Synthesis of Lipophilic, Phosphoramidate d4T-MP Prodrugs Expressing High Potency Against HIV in Cell Culture: Structural Determinants for in vitro Activity and QSAR. Siddiqui, A.; McGuigan, C.; Gilbert, I.H.; Ballatore, C.; Zuccotto, F.; De Clercq, E.; Balzarini, J. J. Med. Chem., 1999,42, 4122-4128.\u00a0 \"link<\/a>\u00a0 \"link<\/a><\/p>\n

Inhibitors of Protease-Resistant Prion Formation. Gilbert I. H.; Rudyk, H.; International Antiviral News, 1999, 7, 78-82.<\/p>\n

The Structure-Based Design And Synthesis Of Selective Inhibitors of Trypanosoma cruzi Dihydrofolate Reductase. Zuccotto, F.; Brun, R.; Gonzalez Pacanowska, D.; Ruiz Perez, L. M.; Gilbert, I. H. Bioorg. Med. Chem. Lett., 1999, 9, 1463-1468.\u00a0 \"link<\/a>\u00a0 \"link<\/a><\/p>\n

General Synthesis of 3-Phosphorylated myo-Inositol Phospholipids and their Derivatives. Painter, G. F.; Grove, S. J. A.; Gilbert, I. H.; Holmes, A. B.; Raithby, P. R.; Hill, M. L.; Hawkins, P. T.; Stephens, L. R. J. Chem. Soc., Perk. T 1, 1999, 923-936.\u00a0 \"link<\/a><\/p>\n

Design And Synthesis Of Bio-Isosteres Of Thymidine Triphosphate. Goldring, A. O.; Balzarini, J.; Gilbert, I. H. Bioorg. Med. Chem. Lett., 1998, 8, 1211-1215.\u00a0 \"link<\/a>\u00a0 \"link<\/a><\/p>\n

An Approach To Use An Unusual Adenosine Transporter To Selectively Deliver Polyamine Analogues To Trypanosomes. Tye, C.-K.; Kasinathan, G.; Barrett, M. P.; Brun, R.; Doyle, V. E.; Fairlamb, A. H.; Weaver R.; Gilbert, I. H. Bioorg. Med. Chem. Lett., 1998, 8, 811-816.\u00a0 \"link<\/a>\u00a0 \"link<\/a><\/p>\n

Electrospray Mass Spectrometry For Assay of Erythromycin A Extracted From Fermentation Liquor. Morgan, J.; Rowlands, R. T.; Joyce-Menekse, M. E.; Gilbert, I. H.; Lloyd, D. Biotechnol. Tech., 1998, 12, 435-438.\u00a0 \"link<\/a><\/p>\n

Dihydrofolate Reductase: a Potential Drug Target in Trypanosomes and Leishmania. Zuccotto, F.; Martin, A. C. R.; Laskowski, R. A.; Thornton, J. M.; Gilbert, I. H. J. Comput. Aid. Mol. Des., 1998, 12, 241-257.\u00a0 \"link<\/a>\u00a0 \"link<\/a><\/p>\n

Versatile Synthesis of myo-Inositol Phospholipid Precursors. Grove, S. J. A.; Gilbert, I. H.; Holmes, A. B.; Painter, G. F.; Hill, M. L. Chem. Commun., 1997, 1633-1634.\u00a0 \"link<\/a><\/p>\n

The Design and Synthesis of Nucleoside Triphosphate Isosteres as Potential Inhibitors of HIV Reverse Transcriptase. R. Weaver, I. H. Gilbert, Tetrahedron, 1997, 53, 5537-5562.\u00a0 \"link<\/a><\/p>\n

Lipophilic Bioisosteres of Nucleoside Triphosphates. Goldring, A. O.; Gilbert, I. H.; Mahmood, N.; Balzarini, J. Bioorg. Med. Chem. Lett., 1996, 6, 2411-2416.\u00a0 \"link<\/a><\/p>\n

Isosteres of Nucleoside Triphosphates. Weaver, R.; Gilbert, I. H.; Mahmood, N.; Balzarini, J. Bioorg. Med. Chem. Lett., 1996, 6, 2405-2410.<\/p>\n

Synthesis of \u03b2 -Keto and \u03b1\u03b2 -Unsaturated N-Acetylcysteamine Thioesters. Gilbert, I. H.; Ginty, M.; O’Neill, J. A.; Simpson, T. J.; Staunton J.; Willis C. L. Bioorg. Med. Chem. Lett, 1995, 5, 1587-1590.<\/p>\n

Imidazolines as Amide Bond Replacements. Gilbert, I. H.; Rees, D. C.; Crockett, A. K.; Jones, R. C. F. Tetrahedron, 1995, 51, 6315-6335.\u00a0 \"link<\/a><\/p>\n

Synthesis of a Homochiral Alpha, Alpha-Disubstituted Alpha, Beta-Diamino-Acid. Jones, R. C. F.; Crockett, A. K.; Rees D. C.; Gilbert, I. H.\u00a0 Tetrahedron-Asymmetr., 1994, 5, 1661-1664.<\/p>\n

Lewis Acid Catalysed rearrangements of myo-inositol orthoformate derivatives. Gilbert, I. H.\u00a0 Holmes, A. B.; Pestchanker, M. J.; Young, R. C. Carbohyd. Res., 1992, 234, 117-130.\u00a0 \"link<\/a><\/p>\n

Amide bond replacements: incorporation of a 2,5,5-trisubstituted imidazoline into dipeptides and into a CCK-4 derivative. Gilbert, I. H.; Rees, D. C.; Richardson, R. S. Tetrahedron Lett., 1991, 32, 2277-2280.\u00a0 \"link<\/a><\/p>\n

Synthesis of Protected myo-Inositols. Gilbert, I. H.; Holmes, A. B.; Young, R. C. Tetrahedron Lett., 1990, 31, 2633-2634.<\/p>\n","protected":false},"excerpt":{"rendered":"

Design, Synthesis and Evaluation of Inhibitors of Trypanosomal and Leishmanial Dihydrofolate Reductase. Chowdhury, S. F.; Bernier Villamor, V.; Hurtado Guerrero, R.; Leal, I.; Brun, R.; Croft, S. L.; Goodman, J. M.; Maes, L.; Ruiz-Perez, L. M.; Gonzalez Pacanowska, D.; Gilbert, I. H. J. Med. Chem., 1999, 42 , 4300-4312.\u00a0 \u00a0 The Design and Synthesis of […]<\/p>\n","protected":false},"author":8,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"full-width-page.php","meta":{"footnotes":""},"class_list":["post-704","page","type-page","status-publish","hentry"],"blocksy_meta":[],"_links":{"self":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/704","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/users\/8"}],"replies":[{"embeddable":true,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/comments?post=704"}],"version-history":[{"count":1,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/704\/revisions"}],"predecessor-version":[{"id":1019,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/704\/revisions\/1019"}],"wp:attachment":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/media?parent=704"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}