{"id":70,"date":"2013-09-05T16:57:56","date_gmt":"2013-09-05T16:57:56","guid":{"rendered":"http:\/\/blog.dundee.ac.uk\/ian-gilbert\/?page_id=70"},"modified":"2015-02-16T08:51:15","modified_gmt":"2015-02-16T08:51:15","slug":"papers2010","status":"publish","type":"page","link":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/papers2010\/","title":{"rendered":"Papers 2010"},"content":{"rendered":"

Acetazolamide-based fungal chitinase inhibitors. Schuettelkopf, A.; Gros, L.; Blair, D. E.; Frearson, J. A.; van Aalten, D. M. F.; Gilbert, I. H. Bioorg. Med. Chem. 2010, 18, 8334-8340.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n

Potential application of thymidylate kinase in nucleoside analogue activation in Plasmodium falciparum. Cui, H.; Ruiz-Perez, L. M.; Gonzalez-Pacanowska, D.; Gilbert, I. H. Bioorg. Med. Chem., 2010, 18, 7302-7309.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n

Exploring new inhibitors of Plasmodium falciparum purine nucleoside phosphorylase. Cui, H.; Ruda, G.-F.; Carrero-Lerida, J.; Ruiz-Perez, L. M.; Gilbert, I. H.; Gonzalez-Pacanowska, D. Eur. J. Med. Chem. 2010, 45, 5140-5149.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n

Design and Preparation of Sterol Mimetics as Potential Antiparasitics. Gigante, F.; Kaiser, M.; Brun, R.; Gilbert, I. H. Bioorg. Med. Chem. 2010, 18, 7291-7301.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n

Aryl Phosphoramidates of 5-Phospho Erythronohydroxamic Acid, A New Class of Potent Trypanocidal Compounds. Ruda, G.-F.; Wong, P. E.; Alibu, V. P.; Norval, S.; Read, K. D.; Barrett, M. P.; Gilbert, I. H. J. Med. Chem.; 2010, 53, 6071-6078.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n

Selective delivery of 2-hydroxy APA to Trypanosoma brucei using the melamine motif. Klee, N.; Wong, P. E.; Baragana, B.; El Mazouni, F.; Phillips, M. A.; Barrett, M. P.; Gilbert, I. H. Bioorg. Med. Chem., 2010, 20, 4364-4366.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n

Virtual Fragment Screening for Novel Inhibitors of 6-Phosphogluconate Dehydrogenase. Ruda, G. F.; Campbell, G.; Alibu, V. P.; Barrett, M. P.; Brenk, R.; Gilbert, I. H. Bioorg. Med. Chem., 2010, 18, 5056-5062.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/p>\n

N-myristoyltransferase inhibitors as new leads to treat sleeping sickness. Frearson, J. A.; Brand, S.; McElroy, S. P.; Cleghorn, L. A. T.; Smid, O.; Stojanovski, L.; Price, H. P.; Guther, M. L. S.; Torrie, L. S.; Robinson, D. A.; Hallyburton, I.; Mpamhanga, C. P.; Brannigan, J. A.; Wilkinson, A. J.; Hodgkinson, M.; Hui, R.; Qiu, W.; Raimi, O. G.; Van Aalten, D. M. F.; Brenk, R.; Gilbert, I. H.; Read, K. D.; Fairlamb, A. H.; Ferguson, M. A. J.; Smith, D. F.; Wyatt, P. G. Nature, 2010, 464, 728-732.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n

Structural basis for the efficient phosphorylation of AZTMP and dGMP by Plasmodium falciparum type I thymidylate kinase. Whittingham, J.; Carrero-Lerida, J.; Brannigan, J. A.; Ruiz-Perez, L. M.; Silva, A. P. G.; Fogg, M. J.; Wilkinson, A. J.; Gilbert, I. H.; Wilson, K. S.; Gonzalez-Pacanowska, D. Biochem. J., 2010, 428, 499-509.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n

Water-soluble polymer\u2013drug conjugates for combination chemotherapy against visceral leishmaniasis. Nicoletti, S.; Seifert, K.; Gilbert, I. H. Bioorg. Med. Chem., 2010, 18, 2559\u20132565.\u00a0\u00a0 \"pubmed\"<\/a>\u00a0 \"journal\"<\/a><\/p>\n","protected":false},"excerpt":{"rendered":"

Acetazolamide-based fungal chitinase inhibitors. Schuettelkopf, A.; Gros, L.; Blair, D. E.; Frearson, J. A.; van Aalten, D. M. F.; Gilbert, I. H. Bioorg. Med. Chem. 2010, 18, 8334-8340.\u00a0\u00a0 \u00a0 Potential application of thymidylate kinase in nucleoside analogue activation in Plasmodium falciparum. Cui, H.; Ruiz-Perez, L. M.; Gonzalez-Pacanowska, D.; Gilbert, I. H. Bioorg. Med. Chem., 2010, […]<\/p>\n","protected":false},"author":8,"featured_media":0,"parent":0,"menu_order":4,"comment_status":"closed","ping_status":"closed","template":"full-width-page.php","meta":{"footnotes":""},"class_list":["post-70","page","type-page","status-publish","hentry"],"blocksy_meta":[],"_links":{"self":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/70","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/users\/8"}],"replies":[{"embeddable":true,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/comments?post=70"}],"version-history":[{"count":1,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/70\/revisions"}],"predecessor-version":[{"id":1028,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/70\/revisions\/1028"}],"wp:attachment":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/media?parent=70"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}