{"id":46,"date":"2013-09-05T16:45:49","date_gmt":"2013-09-05T16:45:49","guid":{"rendered":"http:\/\/blog.dundee.ac.uk\/ian-gilbert\/?page_id=46"},"modified":"2015-02-16T08:51:09","modified_gmt":"2015-02-16T08:51:09","slug":"papers-2012","status":"publish","type":"page","link":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/papers-2012\/","title":{"rendered":"Papers 2012"},"content":{"rendered":"<p>Synthesis and Evaluation of \u03b1-Thymidine Analogues as Novel Antimalarials. Cui, H.; Carrero-L\u00e9rida, J.; Silva, A. P.; Whittingham, J. L.; Brannigan, J. A.; Ruiz-P\u00e9rez, L. M.; Read, K. D.; Wilson, K. S.; Gonz\u00e1lez-Pacanowska, D.; Gilbert, I. H. J. Med. Chem., 2012, 55, 10948-10957. \u00a0 <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/23240776\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone\" alt=\"pubmed\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" width=\"50\" height=\"20\" \/><\/a>\u00a0 <a href=\"http:\/\/pubs.acs.org\/doi\/abs\/10.1021\/jm301328h\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone\" alt=\"journal\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/journal.jpg\" width=\"54\" height=\"20\" \/><\/a><\/p>\n<p>Automated design of ligands to polypharmacological profiles. Besnard, J.; Ruda, G. F.; Setola, V.; Abecassis, K.; Rodriguiz, R. M.; Huang, X. P.; Norval, S.; Sassano, M. F.; Shin, A. I.; Webster, L. A.; Simeons, F. R.; Stojanovski, L.; Prat, A.; Seidah, N. G.; Constam, D. B.; Bickerton, G. R.; Read, K. D.; Wetsel, W. C.; Gilbert, I. H.; Roth, B. L.; Hopkins, A. L. Nature, 2012, 492, 215-220.\u00a0\u00a0 <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/23235874\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" alt=\"pubmed\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" width=\"50\" height=\"20\" \/><\/a>\u00a0 <a href=\"http:\/\/www.nature.com\/nature\/journal\/v492\/n7428\/full\/nature11691.html\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone\" alt=\"journal\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/journal.jpg\" width=\"54\" height=\"20\" \/><\/a><\/p>\n<p>Whole organism high-content screening by label-free, image-based bayesian classification for parasitic diseases. Paveley, R. A.; Mansour, N. R.; Hallyburton, I.; Bleicher, L. S.; Benn, A. E.; Mikic, I.; Guidi, A.; Gilbert, I. H.; Hopkins, A. L.; Bickle, Q. D. PloS Negl. Trop. Dis. 2012, 6, e1762.\u00a0\u00a0 <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/22860151\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" alt=\"pubmed\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" width=\"50\" height=\"20\" \/><\/a>\u00a0 <a href=\"http:\/\/www.plosntds.org\/article\/info%3Adoi%2F10.1371%2Fjournal.pntd.0001762\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone\" alt=\"journal\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/journal.jpg\" width=\"54\" height=\"20\" \/><\/a><\/p>\n<p>Quinol Derivatives as Potential Trypanocidal Agents. Capes, A.; Patterson, S.; Wyllie, S.; Hallyburton, I.; Collie, I. T.; McCarroll, A. J.; Stevens, M. F. G.; Frearson, J. A.; Wyatt, P. G.; Fairlamb, A. H.; Gilbert, I. H. Bioorg. Med. Chem., 2012, 20, 1607-1615. \u00a0 <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/22264753\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" alt=\"pubmed\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" width=\"50\" height=\"20\" \/><\/a>\u00a0<a href=\"http:\/\/www.sciencedirect.com\/science\/article\/pii\/S0968089611010248\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone\" alt=\"journal\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/journal.jpg\" width=\"54\" height=\"20\" \/><\/a><\/p>\n<p>Design, Synthesis and Biological Evaluation of Trypanosoma brucei Trypanothione Synthetase Inhibitors. Spinks, D.; Torrie, L. S.; Thompson, S.; Harrison, J. R.; Frearson, J. A.; Read, K. D.; Fairlamb, A. H.; Wyatt, P. G.; Gilbert, I. H. ChemMedChem, 2012, 7, 95-106.\u00a0\u00a0 <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/22162199\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" alt=\"pubmed\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" width=\"50\" height=\"20\" \/><\/a>\u00a0 <a href=\"http:\/\/onlinelibrary.wiley.com\/doi\/10.1002\/cmdc.201100420\/abstract\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone\" alt=\"journal\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/journal.jpg\" width=\"54\" height=\"20\" \/><\/a><\/p>\n<p>Discovery of a Novel Class of Orally Active Trypanocidal N-Myristoyltransferase Inhibitors. Brand, S.; Cleghorn, L. A. T.; McElroy, S. P.; Robinson, D. A.; Smith, V. C.; Hallyburton, I.; Harrison, J. R.; Norcross, N. R.; Norval, S.; Spinks, S.; Stojanovski, L.; Torrie, L. S.; Frearson, J. A.; Brenk, R.; Fairlamb, A. H.; Ferguson, M. A. J.; Read, K. D.; Wyatt, P. G.; Gilbert, I. H. J. Med. Chem. 2012, 55, 140-152. \u00a0 <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/22148754\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" alt=\"pubmed\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" width=\"50\" height=\"20\" \/><\/a>\u00a0 <a href=\"http:\/\/pubs.acs.org\/doi\/abs\/10.1021\/jm201091t\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone\" alt=\"journal\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/journal.jpg\" width=\"54\" height=\"20\" \/><\/a><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Synthesis and Evaluation of \u03b1-Thymidine Analogues as Novel Antimalarials. Cui, H.; Carrero-L\u00e9rida, J.; Silva, A. P.; Whittingham, J. L.; Brannigan, J. A.; Ruiz-P\u00e9rez, L. M.; Read, K. D.; Wilson, K. S.; Gonz\u00e1lez-Pacanowska, D.; Gilbert, I. H. J. Med. Chem., 2012, 55, 10948-10957. \u00a0 \u00a0 Automated design of ligands to polypharmacological profiles. Besnard, J.; Ruda, G. [&hellip;]<\/p>\n","protected":false},"author":8,"featured_media":0,"parent":0,"menu_order":2,"comment_status":"closed","ping_status":"closed","template":"full-width-page.php","meta":{"footnotes":""},"class_list":["post-46","page","type-page","status-publish","hentry"],"blocksy_meta":[],"_links":{"self":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/46","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/users\/8"}],"replies":[{"embeddable":true,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/comments?post=46"}],"version-history":[{"count":1,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/46\/revisions"}],"predecessor-version":[{"id":1022,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/46\/revisions\/1022"}],"wp:attachment":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/media?parent=46"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}