{"id":1091,"date":"2014-04-16T20:38:36","date_gmt":"2014-04-16T20:38:36","guid":{"rendered":"http:\/\/sites.dundee.ac.uk\/ian-gilbert\/?page_id=1091"},"modified":"2015-02-16T08:33:59","modified_gmt":"2015-02-16T08:33:59","slug":"2014papers","status":"publish","type":"page","link":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/2014papers\/","title":{"rendered":"Papers 2014"},"content":{"rendered":"<p>Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma brucei N-Myristoyltransferase Inhibitors: Idenification and Evaluation of CNS Penetrant Compounds as Potential Treatments for Stage 2 Human African Trypanosomiasis. Brand, S.; Norcorss, N. R.; Thompson, S.; Harrison, J. R.; Smith, V. C.; Robinson, D. A.; Torrie, L. S.; McElroy, S. P.; Hallyburton, I.; Norval, S.; Scullion, P.; Stojanovski, L.; Simeons, F. R. C.; van Aalten, D.; Frearson, J. A.; Fairlamb, A. H.; Ferguson, M. A. J.; Wyatt, P. G.; Gilbert, I. H.; Read, K. D. J. Med. Chem., 2014, 57, 9855-9869. <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/25412409\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone wp-image-19 size-full\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" alt=\"\" width=\"50\" height=\"20\" \/><\/a><\/p>\n<p>Characterisation of a melamino nitroheterocycle as a potential lead for the treatment of human African trypanosomiasis. Giordani, F.; Buschini, A.; Baliani, A.; Kaiser, M.; Brun, R.; Barrett, M. P.; Pellacani, C.; Poli, P.; Gilbert, I. H. Antimicrob. Agents Chemother. 2014, 58, 5747-5757. <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/25022590\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone wp-image-19 size-full\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" alt=\"link to journal abstract in pubmed\" width=\"50\" height=\"20\" \/><\/a><\/p>\n<p>Fragment screening reveals salicylci hydroxamic acid as an inhibitor of Trypanosoma brucei GPI GlcNAc-PI deN-acetylase. Urbaniak, M. D.; Capes, A. S.; Crossman, A.; O\u2019Neill, S.; Thompson, S.; Gilbert, I. H.; Ferguson, M. A. J. Carbohydr. Res., 2014, 387, 54-58. <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/24589444\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone  wp-image-19\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" alt=\"link to journal abstract in pubmed\" width=\"50\" height=\"20\" \/><\/a><\/p>\n<p>Probing the substrate specificity of Trypanosoma brucei GlcNAc-PI de-N-acetylase with synthetic substrate analogues. Capes, A. S.; Crossman, A.; Urbaniak, M. D.; Gilbert, S. H.; Ferguson, M. A.; Gilbert, I. H. Org. Biomol. Chem., 2014, 12, 1919-1934. <a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/24519084\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-19\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" alt=\"link to journal abstract in pubmed\" width=\"50\" height=\"20\" \/><\/a><\/p>\n<p>Target-based drug discovery for human African trypanosomiasis: selection of molecular target and chemical matter. Gilbert, I. H. Parasitology, 2014, 141, 28-36.\u00a0<a href=\"http:\/\/www.ncbi.nlm.nih.gov\/pubmed\/23931634\" target=\"_blank\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-19\" src=\"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-content\/uploads\/sites\/4\/2013\/09\/pubmed.jpg\" alt=\"link to journal abstract in pubmed\" width=\"50\" height=\"20\" \/><\/a><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma brucei N-Myristoyltransferase Inhibitors: Idenification and Evaluation of CNS Penetrant Compounds as Potential Treatments for Stage 2 Human African Trypanosomiasis. Brand, S.; Norcorss, N. R.; Thompson, S.; Harrison, J. R.; Smith, V. C.; Robinson, D. A.; Torrie, L. S.; McElroy, S. P.; Hallyburton, I.; Norval, S.; Scullion, [&hellip;]<\/p>\n","protected":false},"author":8,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"full-width-page.php","meta":{"footnotes":""},"class_list":["post-1091","page","type-page","status-publish","hentry"],"blocksy_meta":[],"_links":{"self":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/1091","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/users\/8"}],"replies":[{"embeddable":true,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/comments?post=1091"}],"version-history":[{"count":8,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/1091\/revisions"}],"predecessor-version":[{"id":1203,"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/pages\/1091\/revisions\/1203"}],"wp:attachment":[{"href":"https:\/\/sites.dundee.ac.uk\/ian-gilbert\/wp-json\/wp\/v2\/media?parent=1091"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}